BMX-IN-1 - CAS# 1431525-23-3 0268 Formula: C12H16N4O7

Formula: C12H16N4O7

3 nM in a radioactive enzyme assay and is over 100-fold selective for other histone methyltransferases/HMTs

once-daily oral NS5A inhibitor for the treatment of hepatitis C virus infection

InChiKey: GYLDXIAOMVERTK-UHFFFAOYSA-N

10]phenanthroline

BMX-IN-1 - CAS# 1431525-23-3 0268 Formula: C12H16N4O7BMX IN 1 is a selective irreversible BMX inhibitor for prostate cancer. BMX IN 1 can covalently modifies Cys496. BMX IN 1 inhibits the proliferation of Tel BMX transformed Ba F3 cells at two digit nanomolar concentrations but requires single digit micromolar concentrations to inhibit the proliferation of prostate cancer cell lines. MK2206, is able to potentiate BMX inhibitor's antiproliferation efficacy against prostate cancer cells. Product